WDR5-IN-4 TFA

Overview

WDR5-IN-4 TFA (Compound C6) is an inhibitor of the WIN site of chromatin-associated WD repeat-containing protein 5 ( WDR5 ), with a K d of 0.1 nM. WDR5-IN-4 TFA displaces WDR5 from chromatin and decreases the expression of associated genes, causing translational inhibition, nucleolar stress. Anti-cancer activity.

Application

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Product Information

• Catalog No.: HY-111753A
• CAS No.: 2749300-35-2
• Molecular Formula: C27H23Cl2F4N5O3
• Molecular Weight: 612.40
• Purity: 98.04%
• Storage: 4°C, stored under nitrogen, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen, away from moisture)
• Solubility: ≥ 2.5 mg/mL (4.08 mM); Clear solution
• Availability: In-stock

Source

Original product source