LY456066

Overview

LY456066 is a selective non-competitive metabotropic glutamate receptors ( mGluR1 ) antagonist with an IC 50 value of 52.0 nM. LY456066 is effective in rodent models of anxiolysis and nociception. LY456066 reduces hyperalgesia and the amount of licking and flinching following formalin injection, which is promising for research of analgesics for chronic pain.

Application

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Product Information

• Catalog No.: HY-119097
• CAS No.: 338738-66-2
• Molecular Formula: C19H23N3OS
• Molecular Weight: 341.47
• Purity: 99.0%
• Storage: -20°C, protect from light, stored under nitrogen * In solvent : -80°C, 6 months; -20°C, 1 month (protect from light, stored under nitrogen)
• Availability: In-stock

Source

Original product source