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Kinase Inhibitors & Modulators

Inhibitors, activators and modulators of kinases and phosphorylation pathways.

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HY-W674387Nec-34i 2212541-00-7 Nec-34i is an inactive analog structurally similar to Nec-34 ( HY-132203 ). Nec-34i has no effect on RIPK1 kinase...
HY-183909EphB1-IN-2 2097512-73-5 EphB1-IN-2 is a mutant-selective kinase inhibitor of ABL and FGFR4 , with an IC 50 of 14 nM against ABL G321C mutant...
HY-125585Syk-IN-2 1345458-66-3 Syk-IN-2 (Page 78; 35) is a spleen tyrosine kinase ( Syk ) inhibitor.
HY-W7403781,2,3,4-Tetrahydro Staurosporin 220038-19-7 1,2,3,4-Tetrahydrostaurosporine is a derivative of Staurosporine ( HY-15141 ) and an inhibitor of mutant EGFR ( IC...
HY-W100186Win 47338 80047-24-1 Win 47338 (compound 14) is a control compound of inhibitors of the mitotic kinase monopolar spindle MPS1 and Aurora...
HY-W064657Momelotinib dihydrochloride 1380317-28-1 Momelotinib (dihydrochloride) is a JAK1/JAK2 inhibitor that also antagonizes ACVR1 , leading to downregulation of...
HY-W0426484,5,6,7-Tetrabromo-1H-benzimidazole 577779-57-8 4,5,6,7-Tetrabromobenzimidazole is a selective and ATP competitive CK2 ( casein kinase 2) inhibitor.
HY-W0068331-Phenylindole 16096-33-6 1-Phenylindole (Compound 8) is a 1-Phenylbenzimidazole analogue. 1-Phenylindole shows IC 50 values of >50 μM and >50...
HY-W0012195-Bromothiazol-2-amine 3034-22-8 5-Bromothiazol-2-amine (Compound 54) is a simple amino. 5-Bromothiazol-2-amine shows an IC 50 of >10 µM against...
HY-N8724Lamalbid 52212-87-0 Lamalbid is a natural product that can be found in Lantana montevidensis . Lamalbid inhibits ROS generation.
HY-B0794SAZ7550-d 5 2719690-99-8 AZ7550 -d 5 is the deuterium labeled AZ7550 ?( HY-B0794 ). AZ7550 , an active metabolite of Osimtinib (AZD9291...
HY-51327CK1-IN-5 1000340-33-9 CK1-IN-5 (compound B-AZ) is an inhibitor of CK1 . CK1-IN-5 lengthened the circadian period by inhibits AtCKL3/AtCKL4...
HY-49459Casein kinase 1δ-IN-14 793722-88-0 Casein kinase 1δ-IN-14 (compound 481) is a casein kinase inhibitor that can be used to study neurodegenerative...
HY-213363-Azetidinemethanol hydrochloride 928038-44-2 3-Azetidinemethanol hydrochloride, an intermediate, can be used in the synthesis of SHP2 inhibitor .
HY-18958A(S)-CCT245737 1489389-23-2 (S)-CCT245737 ((S)-SRA737) is a potent and selective oral inhibitor of checkpoint kinase 1 (CHK1) .
HY-18651(E/Z)-Rigosertib sodium 1225497-78-8 Rigosertib (ON-01910) is a biochemical reagent that can be used as a biological material or organic compound for...
HY-181754TPKI-39 1005781-50-9 TPKI-39 is a DDR1 , DDR2 , and FLT1 inhibitor, with a human DDR1 IC 50 of 380 nM, human DDR1 K a of 24 nM, human...
HY-181586CK1γ-IN-1 1397706-29-4 CK1γ-IN-1 is a non-selective CK1 kinase inhibitor with IC 50 values of 780 nM, 570 nM and 990 nM against human...
HY-181585FP1-24 1403557-08-3 FP1-24 is a non-selective CK1 kinase inhibitor, with IC 50 values of 40 nM, 10 nM, 10 nM, and 40 nM against human...
HY-181584AKI-062a 1093303-07-1 AKI-062a is a non-selective kinase inhibitor, such as a CK1γ inhibitor. AKI-062a binds to and inhibits WNT pathway...

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