Pimozide -d 5 (R6238-d 5 ) is the deuterium labeled Pimozide ( HY-12987 ). Pimozide is a dopamine receptor antagonist , with Kis of 1.4 nM, 2.5 nM and 588 nM for dopamine D2, D3 and D1 receptors, respectively, and also has affinity at α1-adrenoceptor, with a Ki of 39 nM; Pimozide also inhibits STAT3 and STAT5 .
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