N-Desmethyl apalutamide-d 4

Overview

N-Desmethyl apalutamide-d 4 is the deuterium-labeled N-Desmethyl-Apalutamide ( HY-135331 ). N-Desmethyl Apalutamide is an active metabolite of Apalutamide. N-Desmethyl Apalutamide is a less potent antagonist of the androgen receptor and is responsible for one-third of the activity of Apalutamide. The formation of N-Desmethyl Apalutamide mediated predominantly by CYP2C8 and CYP3A4 . N-Desmethyl Apalutamide is moderate to strong CYP3A4 and CYP2B6 inducer and has an excellent plasma-proteins bound concentration.

Application

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Product Information

• Catalog No.: HY-W754151
• CAS No.: 1332391-11-3
• Molecular Formula: C20H9D4F4N5O2S
• Molecular Weight: 467.43
• Purity: 99.63%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Availability: In-stock

Source

Original product source