TCS 1102

Overview

TCS 1102 is a potent, dual orexin receptor antagonist, with Ki values of 0.2 nM and 3 nM for OX2 and OX1 receptors, respectively. TCS 1102 demonstrates excellent blood-brain barrier penetrability and moderate bioavailability in rats.

Application

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Product Information

• Catalog No.: HY-10900
• CAS No.: 916141-36-1
• Molecular Formula: C27H26N4O2S
• Molecular Weight: 470.59
• Purity: 99.73%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 2 years , -20°C, 1 year
• Solubility: ≥ 2.5 mg/mL (5.31 mM); Clear solution
• Availability: In-stock

Source

Original product source