A 967079

Overview

A 967079 is a selective TRPA1 channel blocker (IC50 = 67 and 289 nM at human and rat TRPA1 receptors, respectively) with 1000-fold selectivity for TRPA1 over other TRP channels. A 967079 was shown to have analgesic effects in a rat osteoarthritic pain model.

Application

Products > Drug Discovery > Inhibitor | Products > Drug Discovery > Inhibitor | Cardiovascular and blood system | TRP Channel

Product Information

• Catalog No.: B0084-359603
• CAS No.: 1170613-55-4
• Molecular Formula: C12H14FNO
• Molecular Weight: 207.24
• Purity: ≥98% by HPLC

Source

Original product source