Afatinib dimaleate

Afatinib dimaleate
  • CAS No.:850140-73-7
  • Grade:>98%
  • Formula:C32H33ClFN5O11
  • M.W.:717.18

Overview

Afatinib Dimaleate irreversibly inhibits EGFR/HER2 including EGFR(wt), EGFR(L858R), EGFR(L858R/T790M) and HER2 with IC50 of 0.5 nM, 0.4 nM, 10 nM and 14 nM, respectively.

Application

Products > Drug Discovery > Impurities > Anti-Neoplastic > Afatinib and Impurities | Products > Drug Discovery > Inhibitor

Product Information

  • Catalog No.: B0084-463336
  • CAS No.: 850140-73-7
  • Molecular Formula: C32H33ClFN5O11
  • Molecular Weight: 717.18
  • Purity: >98%

Source

Original product source


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