SB705498

Overview

SB705498 is a TRPV1 antagonist for hTRPV1, antagonizes capsaicin, acid, and heat activation of TRPV1 with IC50 of 3 nM, 0.1 nM and 6 nM, shows a degree of voltage dependence, exhibits >100-fold selectivity for TRPV1 over TRPM8.

Application

Products > Drug Discovery > Inhibitor | Products > Drug Discovery > Inhibitor | Cardiovascular and blood system | TRP Channel

Product Information

• Catalog No.: B2693-453478
• CAS No.: 501951-42-4
• Molecular Formula: C17H16BrF3N4O
• Molecular Weight: 429.23
• Purity: >98%

Source

Original product source