PD176252 (Standard)

Overview

PD176252 (Standard) is the analytical standard of PD176252 ( HY-103286 ). This product is intended for research and analytical applications. PD176252 is a potent antagonist of neuromedin-B preferring (BB1) and gastrin-releasing peptide-preferring (BB2) receptor with Kis of 0.17 nM and 1 nM for human BB1 and BB2 receptors, and 0.66 nM, 16 nM for Rat BB1 and BB2 receptors, respectively; PD176252 is also an agonist of N-Formyl peptide receptor1/2 (FPR1/FPR2), with EC 50 s of 0.31 and 0.66 μM in HL-60 cells.

Application

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Product Information

• Catalog No.: HY-103286R
• CAS No.: 204067-01-6
• Molecular Formula: C32H36N6O5
• Molecular Weight: 584.67
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source