SB-657510 (Standard)

Overview

SB-657510 (Standard) is the analytical standard of SB-657510 ( HY-10656 ). This product is intended for research and analytical applications. SB-657510 is a selective urotensin II (UII) receptor (UT) antagonist. The K i values are 61, 17, 30, 65 and 56 nM for human, monkey, cat, rat and mouse receptors, respectively. SB-657510 exerts anti-inflammatory effects by inhibiting UII-induced upregulation of inflammatory mediators such as adhesion molecules, cytokines, and tissue factor in human vascular endothelial cells.

Application

Products | Products > Signaling Pathways > Others | Products > Signaling Pathways > GPCR/G Protein | Products > Research Areas > Inflammation/Immunology | Products > Signaling Pathways > Reference Standards | Products > Signaling Pathways > Urotensin Receptor

Product Information

• Catalog No.: HY-10656R
• CAS No.: 474960-44-6
• Molecular Formula: C19H22BrClN2O5S
• Molecular Weight: 505.81
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source