RHC 80267 (Standard) is the analytical standard of RHC 80267 ( HY-107416 ). This product is intended for research and analytical applications. RHC 80267 (U-57908) is a potent and selective inhibitor of diacylglycerol lipase ( DAGL ) (with IC 50 of 4 μM in canine platelets). RHC-80267 inhibits cholinesterase activity with an IC 50 of 4 μM, thereby enhancing the relaxation evoked by acetylcholine. RHC 80267 also inhibits COX and the hydrolysis of phosphatidylcholine (PC).
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