Opiranserin hydrochloride (Standard)

Overview

Opiranserin hydrochloride (Standard) is the analytical standard of Opiranserin (hydrochloride) ( HY-109067A ). This product is intended for research and analytical applications. Opiranserin (VVZ-149) hydrochloride, a non-opioid and non-NSAID analgesic candidate, is a dual antagonist of glycine transporter type 2 ( GlyT2 ) and serotonin receptor 2A (5HT2A), with IC 50 s of 0.86 and 1.3 μM, respectively. Opiranserin hydrochloride shows antagonistic activity on rP2X3 (IC 50 =0.87 μM). Opiranserin hydrochloride is development as an injectable agent for the treatment of postoperative pain.

Application

Products | Products > Signaling Pathways > Others | Products > Signaling Pathways > Membrane Transporter/Ion Channel | Products > Signaling Pathways > Neuronal Signaling | Products > Signaling Pathways > GPCR/G Protein | Products > Research Areas > Neurological Disease | Products > Signaling Pathways > Reference Standards | Products > Signaling Pathways > GlyT | Products > Signaling Pathways > 5-HT Receptor | Products > Signaling Pathways > P2X Receptor

Product Information

• Catalog No.: HY-109067AR
• CAS No.: 1440796-75-7
• Molecular Formula: C21H35ClN2O5
• Molecular Weight: 430.97
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source