CHF-2993 is an orally active anticonvulsant. CHF-2993 antagonizes Bicuculline ( HY-N0219 )- and Picrotoxin (HY-101391)-induced tonic convulsions in mice, shows no activity against Pentylenetetrazole-induced clonic convulsions in mice, and partially reduces Veratridine ( HY-N6691 )-induced aspartate efflux in rat cortical synaptosomes. CHF-2993 can be used in the research of epilepsy.
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