Lerimazoline

Lerimazoline
  • CAS No.:54765-26-3
  • Formula:C13H18N2
  • M.W.:202.30

Overview

Lerimazoline is a selective 5-HT1D receptor agonist with K i values of 72 and 3480 nM for h5-HT1D and h5-HT1B . Lerimazoline inhibits Forskolin ( HY-15371 )-stimulated cAMP production and induces contractions in rabbit saphenous vein preparations. Lerimazoline can be used for the research of migraine.

Application

Products | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Disease Areas > Blood or Cardio-cerebrovascular Disease | Products > Disease Areas > Pain | Products > Disease Areas > Migraine | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Cardiovascular Disease | Products > Research Areas > Neurological Disease | Products > Signaling Pathways > 5-HT Receptor

Product Information

  • Catalog No.: HY-135079
  • CAS No.: 54765-26-3
  • Molecular Formula: C13H18N2
  • Molecular Weight: 202.30
  • Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source


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