Lerimazoline is a selective 5-HT1D receptor agonist with K i values of 72 and 3480 nM for h5-HT1D and h5-HT1B . Lerimazoline inhibits Forskolin ( HY-15371 )-stimulated cAMP production and induces contractions in rabbit saphenous vein preparations. Lerimazoline can be used for the research of migraine.
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