RTICBM-74

Overview

RTICBM-74 is a blood-brain barrier-permeable, selective CB1 allosteric modulator with IC 50 values of 23 nM (calcium mobilization assay) and 153 nM ([ 35 S]GTPγS assay). RTICBM-74 inhibits CB1 receptor signaling. RTICBM-74 reduces alcohol intake in rats. RTICBM-74 can be used for the research of alcohol use disorder.

Application

Products | Products > Disease Areas > Metabolic or Endocrine Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Research Areas > Metabolic Disease | Products > Signaling Pathways > Cannabinoid Receptor

Product Information

• Catalog No.: HY-182697
• CAS No.: 2130881-32-0
• Molecular Formula: C19H14ClFN2O
• Molecular Weight: 340.78
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source