Lapatinib - 13 C,d 7 (GW572016- 13 C,d 7 ) is the deuterium and 13 C-labeled Lapatinib ( HY-50898 ). Lapatinib (GW572016) is a potent, orally active inhibitor of the ErbB-2 and EGFR tyrosine kinase domains with IC 50 values against purified EGFR and ErbB-2 of 10.2 and 9.8 nM, respectively.
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