AZ-5104 is an active, demethylated metabolite of AZD 9291. AZ-5104 is an EGFR inhibitor with IC 50 s of 1, 6, 1, 25 and 7 nM for EGFR L858R/T790M , EGFR L858R , EGFR L861Q , EGFR and ErbB4, respectively.
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