Tucatinib

Tucatinib
  • CAS No.:937263-43-9
  • Formula:C26H24N8O2
  • M.W.:480.5

Overview

Tucatinib acts as an HER2 inhibitor, and in BT474 breast carcinoma cells, it effectively suppresses HER2 phosphorylation. Tucatinib inhibits AKT phosphorylation and induces apoptosis in BT474 cells, rendering it a viable cytotoxic agent for formulating antibody-drug conjugates (ADCs).

Application

Products > ADC Linker, ADC Payload > ADC Payload | Products > ADC Linker, ADC Payload > ADC Payload > Tucatinib

Product Information

  • Catalog No.: BP-40974
  • CAS No.: 937263-43-9
  • Molecular Formula: C26H24N8O2
  • Molecular Weight: 480.5
  • Storage: -20°C
  • Availability: 24 Hours

Source

Original product source


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