H4R antagonist 1

Overview

H4R antagonist 1 is a potent and highly selective histamine H4 receptor ( H4R ) antagonist with an IC 50 of 27 nM. H4R antagonist 1 does not show any noticeable binding affinity to other subtypes of histamine receptors, H1R, H2R, and H3R.

Application

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Product Information

• Catalog No.: HY-111501
• CAS No.: 1429375-54-1
• Molecular Formula: C11H11BrN8
• Molecular Weight: 335.16
• Purity: 99.82%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2 mg/mL (5.97 mM); Clear solution
• Availability: In-stock

Source

Original product source