TAK-828F

Overview

TAK-828F is a potent, selective, and orally available retinoic acid receptor-related orphan receptor γt ( RORγt ) inverse agonist (binding IC 50 =1.9 nM, reporter gene IC 50 =6.1 nM). TAK-828F shows excellent RORγt isoforms selectivity (>5000-fold selectivity against human RORα and RORβ ).

Application

Products | Products > Disease Areas > Inflammation or Immune System Disease | Products > Signaling Pathways > Metabolic Enzyme/Protease | Products > Signaling Pathways > Vitamin D Related/Nuclear Receptor | Products > Research Areas > Inflammation/Immunology | Products > Signaling Pathways > ROR

Product Information

• Catalog No.: HY-111509
• CAS No.: 1854901-94-2
• Molecular Formula: C28H32FN3O5
• Molecular Weight: 509.57
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source