GSK 5959

Overview

GSK-5959 CAS:901245-65-6 is a potent, selective and cell-permeable BRPF1 bromodomain inhibitor with IC50 ~80 nM. More than 100-fold selectivity for BRPF1 (IC50 = 80 nM) over other 35 bromodomains including BRPF2/3 and BET family bromodomains.

Application

Polyethylene Glycol PEG Linkers > PROTAC Linker > BET Inhibitors

Product Information

• Catalog No.: AP14260
• CAS No.: 901245-65-6
• Molecular Formula: C22H26N4O3
• Molecular Weight: 394.50
• Purity: ≥95%
• Availability: In Stock

Source

Original product source