GSK 2801

Overview

GSK2801 is a selective, cell-permeable inhibitor of the BAZ2 family of bromodomain-containing proteins. GSK 2801 is selective for BAZ2A and BAZ2B inhibitors, with Kd values of 0.26 and 0.14 µM (IC50 values are 0.40 and 0.43 μM), respectively. GSK2801 does not interact with the bromodomains of BRD4(BD1), CREBBP, TRIM24/TIF1α, PB1(BD5), PCAF, or ATAD2. Please contact us for GMP-grade inquiries.

Application

Products > PROTAC, Molecular glue > Inhibitors

Product Information

• Catalog No.: BP-25352
• CAS No.: 1619994-68-1
• Molecular Formula: C20H21NO4S
• Molecular Weight: 371.5
• Storage: -20°C
• Availability: In Stock

Source

Original product source