Homo-PROTAC cereblon degrader 1

Homo-PROTAC cereblon degrader 1
  • CAS No.:2244520-98-5
  • Grade:99.66%
  • Formula:C32H32N6O10
  • M.W.:660.63
  • Solvent:≥ 5 mg/mL (7.57 mM); Clear solution

Overview

Homo-PROTAC cereblon degrader 1 (compound 15a) is a highly potent and efficient Cereblon ( CRBN ) degrader with only minimal effects on IKZF1 and IKZF3 . (Pink: Cereblon ligand ( HY-10984 ); Blue: Cereblon ligand ( HY-10984 ); Black: linker ( HY-W017440 )).

Application

Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > PROTAC | Products > Research Areas > Cancer | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Signaling Pathways > PROTACs

Product Information

  • Catalog No.: HY-111594
  • CAS No.: 2244520-98-5
  • Molecular Formula: C32H32N6O10
  • Molecular Weight: 660.63
  • Purity: 99.66%
  • Storage: 4°C, stored under nitrogen * In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen)
  • Solubility: ≥ 5 mg/mL (7.57 mM); Clear solution
  • Availability: In-stock

Source

Original product source


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