GSK 5959

Overview

GSK 5959 exhibits >100-fold selectivity for BRPF1 (IC50 = 80 nM) over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Inhibits BRPF1 interaction with histone H3.3, which is involved in the epigenetic regulation of gene expression. Please contact us for GMP-grade inquiries.

Application

Products > PROTAC, Molecular glue > Inhibitors

Product Information

• Catalog No.: BP-25353
• CAS No.: 901245-65-6
• Molecular Formula: C22H26N4O3
• Molecular Weight: 394.5
• Storage: -20°C
• Availability: In Stock

Source

Original product source