Endo-BCN-PEG4-Val-Cit-PAB-MMAE is a cutting-edge cleavable linker for ADCs, featuring Val-Cit for selective cleavage by cathepsin B and a potent MMAE payload that targets and kills cancer cells by disrupting microtubules.
Polyethylene Glycol PEG Linkers > Peptide Linkers > Val-Cit Linker
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