VU0529331

Overview

VU0529331 is a homomeric GIRK channel activator, with an EC 50 value of 5.1 μM for human GIRK2 and an EC 50 value of 22.3 μM for GIRK4 . VU0529331 serves as a starting point for the development of non- GIRK1 /X channel probes and also acts as a tool for studying homomeric GIRK channels. VU0529331 is applicable to research related to addiction, primary aldosteronism and delayed-onset obesity.

Application

Products | Products > Disease Areas > Metabolic or Endocrine Disease | Products > Disease Areas > Neurological, Eye or Ear Disease | Products > Disease Areas > Lipid Metabolism | Products > Disease Areas > Obesity | Products > Signaling Pathways > Membrane Transporter/Ion Channel | Products > Research Areas > Neurological Disease | Products > Research Areas > Metabolic Disease | Products > Signaling Pathways > Potassium Channel

Product Information

• Catalog No.: HY-112705
• CAS No.: 1286725-49-2
• Molecular Formula: C22H20N6O
• Molecular Weight: 384.43
• Purity: 99.81%
• Storage: Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 1.25 mg/mL (3.25 mM); Clear solution
• Availability: In-stock

Source

Original product source