Cibenzoline succinate (Cifenline succinate) is the succinate form of Cibenzoline ( HY-106577 ). Cibenzoline succinate is an inhibitor for ATP-sensitive potassium ( KATP ) channel by affecting the pore-forming Kir6.2 subunit with IC 50 of 22.2 µM. Cibenzoline succinate affects insulin secretion and exhibits antiarrhythmic and antidiabetic activities.
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