BMS711939 is a selective agonist for peroxisome proliferator-activated receptor α ( PPAR α ), with EC 50 of 4 nM and 4.5 μM, for human PPARα and human PPARγ . BMS711939 exhibits good pharmacokinetic characters in rats models. BMS711939 increases HDL cholesterol , reduces LDL cholesterol and triglycerides.
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