OPC-14523 hydrochloride

Overview

OPC-14523 hydrochloride is an orally active sigma and 5-HT1A receptor agonist, with high affinity for sigma receptors (σ1/2 IC 50 =47/56 nM), the 5-HT1A receptor ( IC 50 =2.3 nM), and the 5-HT transporter ( IC 50 =80 nM). OPC-14523 hydrochloride shows antidepressant-like activity.

Application

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Product Information

• Catalog No.: HY-116594A
• CAS No.: 145969-31-9
• Molecular Formula: C23H29Cl2N3O2
• Molecular Weight: 450.40
• Purity: 99.95%
• Storage: 4°C, sealed storage, away from moisture * In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
• Solubility: ≥ 2.08 mg/mL (4.62 mM); Clear solution
• Availability: In-stock

Source

Original product source