Zacopride is an orally active 5-HT 3 receptor ( K i of 0.38 nM) antagonist and 5-HT 4 receptor ( K i of 373 nM) agonist. Zacopride exhibits multiple activities, such as regulating gastrointestinal motility, affecting cardiac function, and exerting anxiolytic and antiemetic effects. Zacopride is currently mainly used in the research of gastrointestinal diseases, cardiovascular diseases, and psychiatric diseases such as anxiety.
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