VU0652925, an analog of BMS986120, is a PAR4 antagonist, with IC 50 values of 43 pM and 39.2 pM for PAC1 and P-selectin , respectively. VU0652925 is able to suppress GPIIbIIIa activation.
Products | Products > Disease Areas > Inflammation or Immune System Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Immunology/Inflammation | Products > Research Areas > Inflammation/Immunology | Products > Signaling Pathways > Protease Activated Receptor (PAR) | Products > Signaling Pathways > P-selectin
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