PROTAC FAK degrader 1

PROTAC FAK degrader 1
  • CAS No.:2301916-69-6
  • Grade:99.25%
  • Formula:C47H56F3N9O8S2
  • M.W.:996.13
  • Solvent:≥ 5 mg/mL (5.02 mM); Suspended solution

Overview

PROTAC FAK degrader 1 (Compound PROTAC-3) is a selective and effective degrader of Fak PROTAC with a DC 50 of 3.0 nM. PROTAC FAK degrader 1 reduces the ability of cancer cells to migrate and invade. PROTAC FAK degrader 1 can be used in the study of tumor. (Pink: FAK ligand ( HY-44146 ); Blue: VHL ligand ( HY-125845 ); Black: linker ( HY-44141 )).

Application

Products | Products > Disease Areas > Cancer | Products > Signaling Pathways > PROTAC | Products > Signaling Pathways > Protein Tyrosine Kinase/RTK | Products > Signaling Pathways > PI3K/Akt/mTOR | Products > Research Areas > Cancer > Cancer Targeted Therapy | Products > Research Areas > Cancer > Cancer Metabolism and Metastasis | Products > Research Areas > Cancer | Products > Signaling Pathways > PROTACs | Products > Signaling Pathways > FAK | Products > Signaling Pathways > Akt

Product Information

  • Catalog No.: HY-119932
  • CAS No.: 2301916-69-6
  • Molecular Formula: C47H56F3N9O8S2
  • Molecular Weight: 996.13
  • Purity: 99.25%
  • Storage: -20°C, stored under nitrogen * In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen)
  • Solubility: ≥ 5 mg/mL (5.02 mM); Suspended solution
  • Availability: In-stock

Source

Original product source


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