Rodatristat

Overview

Rodatristat (KAR5417) is a potent tryptophan hydroxylase 1 (TPH1) and TPH2 inhibitor with IC 50 s value of 33 nM and 7 nM, respectively, and shows robust reduction of intestinal serotonin (5-HT) levels in mice.

Application

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Product Information

• Catalog No.: HY-120083
• CAS No.: 1673568-73-4
• Molecular Formula: C27H27ClF3N5O3
• Molecular Weight: 561.98
• Purity: 98.41%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: 2 mg/mL (3.56 mM); Clear solution; Need ultrasonic
• Availability: In-stock

Source

Original product source