Samelisant

Overview

Samelisant (SUVN-G3031) is a potent and selective histamine H3 receptor (H3R) inverse agonist with good brain penetration and oral bioavailability. Samelisant has a similar binding affinity towards human (hH3R; K i =8.7 nM) and rat (rH3R;K i =9.8 nM) H3R indicating no inter-species differences. Samelisant can be used for the research of sleep-related disorders.

Application

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Product Information

• Catalog No.: HY-120124
• CAS No.: 1394808-20-8
• Molecular Formula: C21H33Cl2N3O3
• Molecular Weight: 446.41
• Purity: 98.65%
• Storage: Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.08 mg/mL (4.66 mM); Clear solution
• Availability: In-stock

Source

Original product source