Orvepitant maleate

Overview

Orvepitant maleate (GW823296 maleate) is potent, selective, orally active and well-tolerated neurokinin-1 receptor (NK-1) antagonist with a pK i of 10.2 for human neurokinin-1 receptor . Orvepitant maleate can across the blood-brain barrier. Orvepitant maleate has the potential for depressive disorder and chronic refractory cough (CRC) treatment.

Application

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Product Information

• Catalog No.: HY-122347A
• CAS No.: 579475-24-4
• Molecular Formula: C35H39F7N4O6
• Molecular Weight: 744.70
• Purity: 99.99%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 5 mg/mL (6.71 mM); Clear solution
• Availability: In-stock

Source

Original product source