Samidorphan

Overview

Samidorphan (ALKS-33) is an orally active opioid system modulator that has a high affinity for binding with μ‐opioid, κ‐opioid, and δ‐opioid receptors. Samidorphan acts as an antagonist at μ‐opioid receptors and acts as a partial agonist at k-opioid and δ‐opioid receptors. Samidorphan primarily acts as an opioid receptor antagonist in vivo. Samidorphan can improve the behavior of depressed animals .

Application

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Product Information

• Catalog No.: HY-123689
• CAS No.: 852626-89-2
• Molecular Formula: C21H26N2O4
• Molecular Weight: 370.44
• Purity: 99.04%
• Storage: Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 5 mg/mL (13.50 mM); Clear solution
• Availability: In-stock

Source

Original product source