Contilisant is a permeable antioxidant and neuroprotectant agent. Contilisant exhibits high nM affinity at H3R . Contilisant inhibits monoamine oxidases and cholinesterases . Contilisant has a binding affinity of 65.23 nM towards hS1R. Contilisant can significantly restore cognitive deficit induced by Aβ 1-42 in the radial maze assay of Alzheimer’s animal model.
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