VU0071063

Overview

VU0071063 is a potent and specific Kir6.2/SUR1 opener ( EC 50 =7.44 μM) and can be used for investigating Kir6.2/SUR1 expressed in the pancreas and brain. VU0071063 inhibits insulin secretion by inducing hyperpolarization of β-cell membrane potential. VU0071063 chemotype has a very steep structure-activity relationships.

Application

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Product Information

• Catalog No.: HY-124424
• CAS No.: 333415-38-6
• Molecular Formula: C18H22N4O2
• Molecular Weight: 326.39
• Purity: 99.71%
• Storage: 4°C, protect from light * In solvent : -80°C, 6 months; -20°C, 1 month (protect from light)
• Solubility: ≥ 2.5 mg/mL (7.66 mM); Clear solution
• Availability: In-stock

Source

Original product source