D13-9001 is a potent AcrB (AcrAB-TolC efflux pump subunit) and MexB (MexAB-OprM efflux pump subunit) inhibitor with the K D values of 1.15 μM and 3.57 μM in E. coli and P. aeruginosa , respectively. D13-9001 exhibits antibiotic activities.
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