Esamisulpride ((S)-Amisulpride) is the S-isomer of Amisulpride ( HY-14545 ). Esamisulpride is a potent dopamine D 2 /D 3 receptor antagonist with K i values of 4.43 nM for D 2 R and 0.72 nM for D 3 R . Esamisulpride is a 5-HT 7 receptor antagonist with a K i of 900 nM. Esamisulpride can be used in the research of schizophrenia and depression.
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