NR2B-selective NMDA receptor antagonist 1

Overview

NR2B-selective NMDA receptor antagonist 1 (compound 29) is a potent antagonist of NR1/NR2B receptors, with IC 50 s of 0.05 μM, 0.73 μM, 2.4 μM to NR1/NR2B NMDA receptor , hERG, α1-AdR, respectivity. NR2B-selective NMDA receptor antagonist 1 exhibites efficient permeability across the blood–brain barrier.

Application

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Product Information

• Catalog No.: HY-126123
• CAS No.: 457897-92-6
• Molecular Formula: C18H22Cl2N2O4S
• Molecular Weight: 433.35
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.
• Availability: In-stock

Source

Original product source