Pimozide-d 5 N-Oxide is the deuterium labeled Pimozide. Pimozide is a dopamine receptor antagonist , with K i s of 1.4 nM, 2.5 nM and 588 nM for dopamine D2, D3 and D1 receptors, respectively, and also has affinity at α1-adrenoceptor, with a Ki of 39 nM; Pimozide also inhibits STAT3 and STAT5 .
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