Theophylline L-lysine (Lysine theophyllinate) is a soluble derivative of Theophylline ( HY-B0809 ). Theophylline L-lysine is a potent phosphodiesterase (PDE) inhibitor, adenosine receptor antagonist, and histone deacetylase ( HDAC ) activator. Theophylline L-lysine inhibits PDE3 activity to relax airway smooth muscle. Theophylline L-lysine has anti-inflammatory activity by increasing IL-10 and inhibiting NF-κB into the nucleus. Theophylline L-lysine induces apoptosis . Theophylline L-lysine can be used for asthma and chronic obstructive pulmonary disease (COPD) research.
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