AdipoR agonist 1 (Compound 112254) is an agonist for adiponectin receptor ( AdipoR ), which activates the transcriptional regulators like peroxisome proliferator-activated receptors (PPARs), peroxisome proliferator-activated receptor gamma coactivator 1α ( PGC-1α ), sirtuin 1 ( SIRT1 ), and adenylate-activated protein kinase ( AMPK ). AdipoR agonist 1 is utilized in preventive doping research.
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