Tubastatin A

Overview

Tubastatin A is a potent and selective HDAC6 inhibitor with an IC 50 of 15 nM in a cell-free assay, and is selective (1000-fold more) against all other isozymes except HDAC8 (57-fold more). Tubastatin A also inhibits HDAC10 and metallo-β-lactamase domain-containing protein 2 (MBLAC2) .

Application

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Product Information

• Catalog No.: HY-13271A
• CAS No.: 1252003-15-8
• Molecular Formula: C20H21N3O2
• Molecular Weight: 335.40
• Purity: 99.07%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 1.25 mg/mL (3.73 mM); Clear solution
• Availability: In-stock

Source

Original product source