(1R,9S)-Exatecan (DX8951) is the (1R,9S) stereoisomer of Exatecan ( HY-13631 ). Exatecan (DX-8951) is a DNA topoisomerase I inhibitor, with an IC 50 of 2.2 μM (0.975 μg/mL), and can be used in cancer research.
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