limertinib

Overview

limertinib (ASK120067) is a potent and orally active inhibitor of EGFR T790M ( IC 50 :0.3 nM) with selectivity over EGFR WT (IC 50 :6.0 nM). limertinib is a third-generation EGFR-TKI for the research of non-small cell lung cancer (NSCLC).

Application

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Product Information

• Catalog No.: HY-138751
• CAS No.: 1934259-00-3
• Molecular Formula: C29H32ClN7O2
• Molecular Weight: 546.06
• Purity: 99.12%
• Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
• Solubility: ≥ 2.5 mg/mL (4.58 mM); Clear solution
• Availability: In-stock

Source

Original product source