Varenicline- 15 N 3 Hydrochloride

Overview

Varenicline-15N3 Hydrochloride (CP 526555-15N3 Hydrochloride) is the 15 N labeled isotope of Varenicline hydrochloride ( HY-10020 ). Varenicline (CP 526555) is an orally active partial agonist of α4β2 nicotinic acetylcholine receptor (α4β2 nAChR , IC 50 = 250 nM), which is the principal mediator of nicotine dependence. Varenicline is also a partial agonist of α6β2 nAChR and a full agonist of α6β2 nAChR . Varenicline blocks the direct agonist effects of nicotine on nAChR while stimulates nAChR in a more moderate way, being widely used as an aid of smoking cessation.

Application

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Product Information

• Catalog No.: HY-10020S
• CAS No.: 1244134-80-2
• Molecular Formula: C13H14Cl15N3
• Molecular Weight: 250.70
• Purity: 99.98%
• Storage: Please store the product under the recommended conditions in the Certificate of Analysis.

Source

Original product source