MCHR1 antagonist 2

MCHR1 antagonist 2
  • CAS No.:863115-70-2
  • Grade:98.27%
  • Formula:C23H21FN2O5
  • M.W.:424.42
  • Solvent:≥ 1 mg/mL (2.36 mM); Clear solution

Overview

MCHR1 antagonist 2 is an antagonist of melanin concentrating hormone receptor 1 , with an IC 50 of 65 nM; MCHR1 antagonist 2 also inhibits hERG , with an IC 50 of 4.0 nM in IMR-32 cells.

Application

Products | Products > Disease Areas > Metabolic or Endocrine Disease | Products > Signaling Pathways > GPCR/G Protein | Products > Signaling Pathways > Neuronal Signaling | Products > Signaling Pathways > Membrane Transporter/Ion Channel | Products > Research Areas > Metabolic Disease | Products > Research Areas > Endocrinology | Products > Signaling Pathways > MCHR1 (GPR24) | Products > Signaling Pathways > Potassium Channel

Product Information

  • Catalog No.: HY-100321
  • CAS No.: 863115-70-2
  • Molecular Formula: C23H21FN2O5
  • Molecular Weight: 424.42
  • Purity: 98.27%
  • Storage: Powder -20°C, 3 years , 4°C, 2 years ; In solvent -80°C, 6 months , -20°C, 1 month
  • Solubility: ≥ 1 mg/mL (2.36 mM); Clear solution
  • Availability: In-stock

Source

Original product source


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